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Research Papers : 2019
A Novel Lead Identification Strategy: Screening an sp
3
-rich and Lead-like Compound Library Composed of 7-Azanorbornane Derivatives.
Karaki, F.; Umemoto, S.; Ashizawa, K.; Sato, N.; Oki, T.; Ogino, T.; Ishibashi, N.; Someya, R.; Miyano, K.; Hirayama, S.; Uezono, Y.; Fujii, H.
ChemMedChem
,
2019
,
14
, 1840-1848.
Ligand-Dependent Site-Selective Suzuki Cross-Coupling of 4-Bromopyrazol-5-yl Triflates.
Sakakibara, R.; Itoh, K.; Fujii, H.
J. Org. Chem.
,
2019
,
84
, 11474-11481.
Development of Novel δ Opioid Receptor Inverse Agonists without a Basic Nitrogen Atom and Their Antitussive Effects in Mice.
Higashi, E.; Hirayama, S.; Nikaido, J.; Shibasaki, M.; Kono, T.; Honjo, A.; Ikeda, H.; Kamei, J.; Fujii, H.
ACS Chem. Neurosci.
,
2019
,
10
, 3939-3945.
THE PRACTICE OF THE SELECTIVE SYNTHETIC METHOD OF ASYMMETRICAL 1,3,5-TRIOXAZATRIQUINANE DERIVATIVES COMPRISED OF THREE DISTINCT CARBONYL COMPOUNDS.
Hirayama, S.; Obayashi, K.; Wada, N.; Ohyama, K.; Fuku, S.; Koyano, K.; Karaki, F.; Itoh, K.; Nagase, H.; Fujii H.
Heterocycles
,
2019
,
99
, 1003-1019.
Discovery of δ Opioid Receptor Full Inverse Agonists and Their Effects on Restraint Stress-induced Cognitive Impairment in Mice.
Hirayama, S.; Iwai, T.; Higashi, E.; Nakamura, M.; Iwamatsu, C.; Itoh, K.; Nemoto, T.; Tanabe, M.; Fujii, H.
ACS Chem. Neurosci.
,
2019
,
10
, 2237-2242.
Novel asymmetric photodimerization reaction of coumarin derivatives bearing a chiral 2-oxazolidinone auxiliary.
Itoh, K.; Odate, F.; Karikomi, T.; Obe, K.; Miyamori, T.; Kamiya, H.; Yoza, K.; Nagai, K.; Fujii, H.; Suga, H.; Tokunaga, K.
RCS Adv.
,
2019
,
9
, 12365-12369.
A facile preparation of functional cycloalkynes via an azide-to-cycloalkyne switching approach.
Yoshida, S.; Kuribara, T.; Ito, H.; Meguro, T.; Nishiyama, Y.; Karaki, F.; Hatakeyama, Y.; Koike, Y.; Kii, I.; Hosoya, T.
Chem. Commun.
,
2019
,
55
, 3556-3559.
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