Publication
Research Papers : 2013年
- The most effective influence of 17-(3-ethoxypropyl) substituent on the binding affinity and the agonistic activity in KNT-127 derivatives, δ opioid receptor agonists
Nemoto, T.; Ida, Y.; Iihara, Y.; Nakajima, R.; Hirayama, S.; Iwai, T.; Fujii, H.; Nagase, H.
Bioorg. Med. Chem., 2013, 21, 7628-7647.
- Design and synthesis of novel opioid ligands with an azabicyclo[2.2.2]octane skeleton having a 7-amide side chain and their pharmacologies
Watanabe, Y.; Kitazawa, S.; Nemoto, T.; Hirayama, S.; Iwai, T.; Fujii, H.; Nagase, H.
Bioorg. Med. Chem., 2013, 21, 3032-3050.
- The effect of 17-N substituents on the activity of the opioid κ receptor in nalfurafine derivatives
Nemoto, T.; Yamamoto, N.; Wada, N.; Harada, Y.; Tomatsu, M.; Ishihara, M.; Hirayama, S.; Iwai, T.; Fujii, H.; Nagase, H.
Bioorg. Med. Chem. Lett., 2013, 23, 268-272.
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