Publication
Research Papers : 2014
- Design, synthesis, and structure–activity relationship of novel opioid κ receptor selective agonists: α-Iminoamide derivatives with an azabicyclo[2.2.2]octene skeleton.
Watanabe, Y.; Kitazawa, S.; Fujii, H.; Nemoto, T.; Hirayama, S.; Iwai, T.; Gouda, H.; Hirono, S.; Nagase, H.
Bioorg. Med. Chem. Lett., 2014, 24, 4980-4983.
- Human nitrilase-like protein does not catalyze the hydrolysis of vildagliptin.
Asakura, M.; Nakano, M.; Hayashida, K.; Fujii, H.; Nakajima, M.; Atsuda, K.; Itoh, T.; Fujiwara, R.
Drug Metab. Pharmacokinet., 2014, 29, 463-469.
- Synthesis of a novel universal opioid receptor agonist with the 1,3,5-trioxazatriquinane skeleton and its pharmacologies.
Hirayama, S.; Wada, N.; Kuroda, N.; Iwai, T.; Yamaotsu, N.; Hirono, S.; Fujii, H.; Nagase, H.
Bioorg. Med. Chem. Lett., 2014, 24, 4895-4898.
- Synthesis and Pharmacology of a Novel κ Opioid Receptor (KOR) Agonist with a 1,3,5-Trioxazatriquinane Skeleton.
Hirayama, S.; Wada, N.; Nemoto, T.; Iwai, T.; Fujii, H.; Nagase, H.; Fujii, H.; Nagase, H.
ACS Med. Chem. Lett., 2014, 5, 868-872.
- Novel Delta Opioid Receptor Agonists with Oxazatricyclodecane Structure.
Fujii, H.; Hayashida, K.; Saitoh, A.; Yokoyama, A.; Hirayama, S.; Iwai, T.; Nakata, E.; Nemoto, T.; Sudo, Y.; Uezono, Y.; Yamada, M.; Nagase, H.; Fujii, H.
ACS Med. Chem. Lett., 2014, 5, 368-372.
- Zinc-Acetic Acid Promoted Reductive Carbon-Nitrogen Bond Cleavage Reaction of α-Aminoketones.
Ishikawa, K.; Tomatsu, M.; Nagase, H.; Fujii, H.
Heterocycles, 2014, 88, 1051-1063.
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