2005
A
facile clay-mediated synthesis of
3,3-diindolyl-2-indolinones from isatins.
Chakrabarty,
M.; Sarkar, S.; Harigaya,
Y.
Journal of Chemical Research, (8), 540-542,
2005.
Total
synthesis of borrelidin. Nagamitsu,
T.;
Harigaya,
Y.;
Ōmura, S. Proceedings of the Japan Academy, Series B:
Physical and Biological Sciences, 81(7), 244-256,
2005.
Determination
of the absolute stereochemistry and asymmetric total
synthesis of madindolines A and B: a practical improvement
to a second-generation approach from the
first-generation. Hirose,
T.; Sunazuka, T.; Yamamoto, D.; Kojima, N.; Shirahata,
T.; Harigaya,
Y.;
Kuwajima, I.; Ōmura, S. Tetrahedron, 61(25),
6015-6039,
2005.
Synthesis
of linear tripeptides for right-hand segments of
complestatin. Yamada,
Y.; Akiba, A.; Arima,
S.;
Okada, C.; Yoshida, K.; Itoh, F.; Kai, T.; Satou, T.;
Takeda, K.; Harigaya,
Y.
Chemical & Pharmaceutical Bulletin, 53(10),
1277-1290,
2005.
Chemical
constituents of Mussaenda incana. Dinda,
B.; Debnath, S.; Majumder, S.; Arima,
S.; Sato,
N.; Harigaya,
Y. Indian
Journal of Chemistry, Section B: Organic Chemistry
Including Medicinal Chemistry, 44B(11), 2362-2366,
2005.
Triterpenoids
from Bignonia unguiscati roots. Dinda,
B.; Utpal, C. D.; Arima,
S.; Sato,
N.; Harigaya,
Y. Indian
Journal of Chemistry, Section B: Organic Chemistry
Including Medicinal Chemistry, 44B(8), 1735-1739,
2005.
Azithromycin
inhibits the formation of flagellar filaments without
suppressing flagellin synthesis in Salmonella enterica
serovar Typhimurium. Matsui,
H.; Eguchi, M.; Ohsumi, K.; Nakamura, A.; Isshiki, Y.;
Sekiya, K.; Kikuchi, Y.; Nagamitsu,
T.;
Masuma, R.; Sunazuka, T.; Ōmura, S. Antimicrobial Agents
and Chemotherapy, 49(8), 3396-3403,
2005.
An
expedient, regioselective synthesis of 2-alkylamino- and
2-alkylthiothiazolo[5,4-e]indoles. Chakrabarty,
M.; Kundu, T.; Arima,
S.;
Harigaya,
Y.
Tetrahedron Letters, 46(16), 2865-2868,
2005.
Absolute
stereochemistries and total synthesis of
(+)/(-)-macrosphelides, potent, orally bioavailable
inhibitors of cell-cell adhesion. Sunazuka,
T.; Hirose, T.; Chikaraishi, N.; Harigaya,
Y.;
Hayashi, M.; Komiyama, K.; Sprengeler, P. A.; Smith III, A.
B.; Ōmura, S. Tetrahedron, 61(15), 3789-3803,
2005.
Preparative
Monohydroxyflavanone Syntheses and a Protocol for Gas
Chromatography-Mass Spectrometry Analysis of
Monohydroxyflavanones. Kagawa,
H.; Shigematsu, A.; Ohta, S.; Harigaya
Y.
Chemical & Pharmaceutical Bulletin., 53(5),
547-554,
2005.
Application
of Intramolecular 1, 3-Dipolar Cyclic Addition of Azide and
Olefin; Construction of (Pyrrolidine-2-ylidene)Glycinate
and Glycinamides. Konda-Yamada,
Y.; Asano, K.; Satou, T.; Monnma, S.; Sakayanagi, M.;
Satou, N.; Takeda, K.; Harigaya,
Y.
Chemical & Pharmaceutical Bulletin, 53(5),
529-536,
2005.
Reaction
of 3/2-formylindoles with TOSMIC: formation of
indolyloxazoles and stable indolyl primary enamines.
Chakrabarty,
M.; Basak, R.; Harigaya,
Y.
Tetrahedron, 61(7), 1793-1801,
2005.
First
isolation of both indolylcarbinols and diindolylalkanes
from microwave-assisted acid (cray)-catalysed reaction of
indols with diethyl ketomalonate. Chakrabarty,
M.; Karmakar, S.; Harigaya,
Y.
Heterocycles, 65(1), 37-48,
2005.
A
γ-lactone
form nafuredin, nafuredin-γ,
also inhibits helminth complex I. Shiomi,
K.; Ui, H.; Suzuki, H.; Hatano, H.; Nagamitsu,
T.;
Takano, D.; Miyadera, H.; Yamashita, T.; Kita, K.; Miyoshi,
H.; Harder, A.; Tomoda, H.; Ōmura, S. Journal of
Antibiotics, 58(1), 50-55,
2005.
Macrolides
with promotive activity of monocyte to macrophage
differentiation. Yoshida,
K.; Sunazuka, T.; Nagai, K.; Sugawara, A.; Cho, A.;
Nagamitsu,
T.;
Harigaya,
Y.;
Otoguro, K.; Akagawa, K.; Ōmura, S. Journal of Antibiotics,
58(1), 79-81,
2005.
A
concise stereoselective route to the indoline spiroaminal
framework of neoxaline and oxaline. Sunazuka,
T.; Shirahata, T.; Tsuchiya, S.; Hirose, T.; Mori,
R.; Harigaya,
Y.;
Kuwajima, I.; Ōmura, S. Organic Letters, 7(5),
941-943,
2005.
Total
synthesis of (-)-physovenine from
(-)-3a-hydroxyfuroindoline. Sunazuka,
T.; Yoshida, K.; Kojima, N.; Shirahata, T.; Hirose, T.;
Handa, M.; Yamamoto, D.; Harigaya,
Y.;
Kuwajima, I.; Ōmura, S. Tetrahedron Letters, 46(9),
1459-1461,
2005.